Patent · US Expired

Benzenesulphonamide compounds

US6589956B2 · kind B2 · utility

1Cited by
3References
13Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 12, 2002
Grant dateJul 8, 2003
Priority date
Expiry dateJul 12, 2022

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D417/14
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A compound of formula (I): wherein:Ra represents a hydroxy, alkoxy, aryloxy or arylalkyloxy group,A represents a CH group or a nitrogen atom, in which case R1 is as defined in the description,or R1—A together represent an oxygen atom or a group, wherein R3 and R4 are as defined in the description,R2 being a hydrogen atom or an alkyl group,Rb and Rc, which may be identical or different, each represents a hydrogen atom, a halogen atom, an alkyl group, an alkoxy group, a hydroxy group or a trihaloalkyl group,n is an integer of from 2 to 6 inclusive,m and p are integers of from 0 to 6 inclusive,its enantiomers, diastereoisomers, and addition salts thereof with a pharmaceutically acceptable acid or base, and medicinal products containing the same which are useful as a TXA2 receptor antagonist and 5-HT2 receptor antagonist.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.