Patent · US Expired

Inhibitors of phospholipase enzymes

US6630496B1 · kind B1 · utility

96Cited by
41References
18Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 24, 2000
Grant dateOct 7, 2003
Priority date
Expiry dateAug 24, 2020

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D417/10
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

This invention provides substituted indole and indoline compounds useful in inhibiting phospholipase activity, particularly including cytosolic phospholipase A2 (cPLA2) activity, as well as pharmaceutical compositions containing the compounds and methods of using them to treat various maladies, including pain and inflammatory conditions.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.