Patent · US Expired

Indolizine SPLA2inhibitors

US6645976B1 · kind B1 · utility

9Cited by
1References
32Claims
0Family size

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Inventors

Key dates

Filing dateApr 28, 1997
Grant dateNov 11, 2003
Priority date
Expiry dateApr 28, 2017

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07F9/6561
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A class of novel indolizine-1-functional compounds and indolizine-3-functional compounds is disclosed together with the use of such indolizine compounds for inhibiting sPLA2 mediated release of fatty acids for treatment of conditions such as septic shock. The compounds are indolizine-1-acetamides, indolizine-1-acetic acid hydrazides, indolizine-1-glyoxylamides, indolizine-3-acetamides, indolizine-3-acetic acid hydraxides, and indolizine-3-glyoxylasides.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.