Patent · US Expired

Carbapenem derivatives

US6677331B2 · kind B2 · utility

2Cited by
3References
24Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 14, 2002
Grant dateJan 13, 2004
Priority date
Expiry dateAug 14, 2022

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P31/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Disclosed is a novel carbapenem derivative having a substituted imidazo[5,1-b]thiazole group at the 2-position on the carbapenem ring have high anti microbial activities against &bgr;-lactamase producing bacteria, MRSA, resistant-Pseudomonas aeruginosa, PRSP, enterococci, and influenza, and high stabilities to DHP-1. According to the present invention, there is provided a compound represented by the formula (I), or a pharmacologically acceptable salt thereof or an ester at the 3-position on the carbapenem ring thereof:

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.