Patent · US Expired

High purity lipopeptides, Lipopeptide micelles and processes for preparing same

US6696412B1 · kind B1 · utility

22Cited by
18References
56Claims
0Family size

Assignee

Inventors

Key dates

Filing dateNov 28, 2000
Grant dateFeb 24, 2004
Priority date
Expiry dateNov 28, 2020

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY10S435/886
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention discloses highly purified daptomycin and to pharmaceutical compositions comprising this compound. The invention discloses a method of purifying daptomycin comprising the sequential steps of anion exchange chromatography, hydrophobic interaction chromatography and anion exchange chromatography. The invention also discloses a method of purifying daptomycin by modified buffer enhanced anion exchange chromatography. The invention also discloses an improved method for producing daptomycin by fermentation of Streptomyces roseosporus. The invention also discloses high pressure liquid chromatography methods for analysis of daptomycin purity. The invention also discloses lipopeptide micelles and methods of making the micelles. The invention also discloses methods of using lipopeptide micelles for purifying lipopeptide antibiotics, such as daptomycin. The invention also discloses using lipopeptide micelles therapeutically.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.