Patent · US Expired

Somatostatin antagonists and agonists that act at the SST subtype 2 receptor

US6696418B1 · kind B1 · utility

14Cited by
1References
23Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 17, 2000
Grant dateFeb 24, 2004
Priority date
Expiry dateJul 17, 2020

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K38/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds according to the formula: and pharmaceutically acceptable salts, solvates or hydrates thereof; wherein group Ar is optionally substituted (C6-C10)aryl or (C1-C9)heteroaryl; X is a direct link, —CH2—, —SO2—, —CO—, —CHR1— where R1 is (C1-C6) alkyl, or —CR1′R1″— where both R1′ and R1″ are, independently, (C1-C6)alkyl; Y is N or CH; and Z and W are as herein defined, and pharmaceutical compositions thereof, and methods useful to facilitate secretion of growth hormone(GH) in mammals.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.