Patent · US Expired

Microbial process for preparing pravastatin

US6750366B2 · kind B2 · utility

5Cited by
4References
2Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 5, 2001
Grant dateJun 15, 2004
Priority date
Expiry dateDec 5, 2021

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC12R2001/645
  • WIPO fieldBiotechnology
  • WIPO sectorChemistry

Abstract

The present invention relates to a new microbial process for the preparation of the compound formula (I): from a compound of general formula (II): wherein R stands for an alkali metal or ammonium ion, by the submerged cultivation of a mold strain able to 6&bgr;-hydroxylate a compound of the Formula (II) in aerobic fermentation and by the separation and purification of the product of Formula (I) formed in the course of the bioconversion. The process comprises cultivating a strain of Mortierella maculata filamentous mold species that is able to 6&bgr;-hydroxylate a compound of the general Formula (II), on a nutrient medium containing assimilable carbon and nitrogen sources and mineral salts and separating the product formed from the fermentation broth, then isolating the compound of formula (I) and purifying the same. Novel strains of Mortierella maculata are also disclosed.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.