Patent · US Expired

7-hexanolytaxol and methods for preparing the same

US6753345B2 · kind B2 · utility

1Cited by
12References
19Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJul 19, 2002
Grant dateJun 22, 2004
Priority date
Expiry dateJul 19, 2022

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P35/02
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

An antitumor compound of formula (5): Also provided by the present invention is a method of preparing a compound of formula (5) whereby diesterification of the alcohol groups located at the 2′ and 7 positions of paclitaxel is followed by the hydrolysis of the 2′ hexanoate group resulting in 7-hexanoyltaxol.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.