Patent · US Expired

Heterocyclic compounds useful as inhibitors of tyrosine kinases

US6770639B2 · kind B2 · utility

189Cited by
4References
22Claims
0Family size

Assignee

Inventors

Key dates

Filing dateNov 12, 2002
Grant dateAug 3, 2004
Priority date
Expiry dateNov 12, 2022

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D513/04
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Disclosed are novel compounds of formula (I): wherein Ar1, Ra, R4, R5, X and Y are defined below, which are useful as inhibitors of certain protein tyrosine kinases and are thus useful for treating diseases associated with such kinases, for example, diseases resulting from inappropriate cell proliferation, which include autoimmune diseases, chronic inflammatory diseases, allergic diseases, transplant rejection and cancer, as well as conditions resulting from cerebral ischemia, such as stroke. Also disclosed are processes for preparing these compounds, novel intermediates useful in these processes and compositions comprising compounds of the formula (I).

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.