Patent · US Expired

Trisubstituted-N-[(1S)-1,2,3,4-Tetrahydro-1-naphthalenyl]benzamides which inhibit P2X3 and P2X2/3 containing receptors

US6831193B2 · kind B2 · utility

2Cited by
0References
68Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 10, 2002
Grant dateDec 14, 2004
Priority date
Expiry dateNov 14, 2022

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D333/72
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Compounds of formula (I) are novel P2X3 and P2X2/P2X3 antagonists which are useful in treating pain, urinary incontinence and bladder overactivity.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.