Patent · US Expired

Fused heteroaryl derivatives

US6838457B2 · kind B2 · utility

44Cited by
5References
19Claims
0Family size

Assignees

Inventors

Key dates

Filing dateJun 10, 2003
Grant dateJan 4, 2005
Priority date
Expiry dateJun 10, 2023

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D495/14
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides a pharmaceutical composition which is useful as a phosphatidylinositol 3 kinase (PI3K) inhibitor and an antitumor agent, and it provides a novel bicyclic or tricyclic fused heteroaryl derivative or a salt thereof which possesses an excellent PI3K inhibiting activity and cancer cell growth inhibiting activity.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.