Glucocorticoid receptor modulators
US6852719B2 · kind B2 · utility
Assignees
Inventors
Key dates
| Filing date | Oct 26, 2001 |
| Grant date | Feb 8, 2005 |
| Priority date | — |
| Expiry date | Oct 26, 2021 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D413/06
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
The present invention provides non-steroidal compounds of Formula I, including prodrugs and pharmaceutically acceptable salts thereof, which are selective modulators (e.g., agonists, partial agonists and antagonists) of a steroid receptor, specifically, the glucocorticoid receptor. The present invention also provides pharmaceutical compositions containing these compounds and methods for using these compounds to treat animals requiring glucocorticoid receptor agonist or antagonist therapy. Glucocorticoid receptor modulators are useful to treat diseases, such as obesity, diabetes, inflammation and others as described below. The present invention also provides processes for preparing these compounds
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.