Patent · US Expired

Combination of benzoquinazoline antifolates and protecting agents

US6855712B2 · kind B2 · utility

1Cited by
4References
1Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 7, 2003
Grant dateFeb 15, 2005
Priority date
Expiry dateNov 22, 2023

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The use of a protecting agent, for example a folate derivative such as folic acid or leucovorin, in combination with a non-competitive folic acid analogue, for example benzoquinazoline derivatives, for use in reducing the side effects associated with the administration of such non-competitive folic acid analogues, and pharmaceutical formulations comprising such combinations are disclosed.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.