Patent · US Expired

Imidazopyrimidine derivatives and triazolopyrimidine derivatives

US6911443B2 · kind B2 · utility

28Cited by
2References
7Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 17, 2001
Grant dateJun 28, 2005
Priority date
Expiry dateApr 17, 2021

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A compound of the formula (I) in which R1 is —OR11, —SR11, —SOR11, —SO2R11, —NHR11, or —NR12R13 , and R11, R12, and R13 are as defined broadly in the text. R2 is H, C1-C6alkyl, carbamoyl, or an ester group. R3 is thienyl, pyridyl optionally substituted by halogen or C1-C6alkoxy; naphthyl optionally substituted by C1-C6alkoxy; dioxane fused phenyl; dioxacyclopentane fused phenyl; or optionally substituted phenyl. Y is CH or N. A process for preparing such compounds, pharmaceutical compositions containing such compounds, and a method of treating asthma using them are also disclosed and claimed.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.