Patent · US Expired

Stable hydrate of a muscarinic receptor antagonist

US6930188B2 · kind B2 · utility

0Cited by
4References
5Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 25, 2003
Grant dateAug 16, 2005
Priority date
Expiry dateApr 16, 2023

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A stable solid hydrate of a muscarinic receptor antagonist is useful in the treatment of irritable bowel syndrome, diverticular disease, oesophageal achalasia, chronic obstructive airways disease, over active bladder (including symptoms of incontinence, urge and frequency), urinary incontinence, neurogenic urinary urgency or pollakiuria, treatment of bladder functional disorder, urinary leakage, painful or difficult urination caused by neurogenic bladder, spastic or hypertonic bladder, dysfunctional bladder syndrome, gastrointestinal disorders including gastrointestinal hyperactivity, and relaxing effect on intestinal smooth muscle cells.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.