Patent · US Expired

Process for producing 2,6-dihalogenopurine

US6936713B2 · kind B2 · utility

2Cited by
2References
16Claims
0Family size

Assignee

Inventors

Key dates

Filing dateApr 3, 2002
Grant dateAug 30, 2005
Priority date
Expiry dateJun 9, 2022

Classification

  • Technology area (CPC Y)Emerging Cross-Sectional Technologies
  • CPC primaryY02P20/55
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A process for conveniently and efficiently preparing a 2,6-dihalogenopurine using an inexpensive starting material. A process for preparing a 2,6-dihalogenopurine, comprising treating a 2-amino-6-halogenopurine having a protective group at 7th position or 9th position with a diazotizating agent and a halogen source; and a process for preparing a 9-acyl-2-amino-6-halogenopurine, comprising treating a 2-amino-6-halogenopurine with an acylating agent in the presence of a base.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.