Patent · US Expired

Methods for isolating crystalline Form I of 5-azacytidine

US6943249B2 · kind B2 · utility

35Cited by
6References
18Claims
0Family size

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Inventors

Key dates

Filing dateMar 17, 2003
Grant dateSep 13, 2005
Priority date
Expiry dateSep 14, 2023

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07H19/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The invention includes methods for isolating crystalline Form I of 5-azacytidine substantially free of other forms, wherein 5-azacytidine is represented by the formula: The invention also includes pharmaceutical compositions comprising Form I of 5-azacytidine.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.