Patent · US Expired

Pharmaceuticals

US6949577B2 · kind B2 · utility

5Cited by
2References
24Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 17, 2003
Grant dateSep 27, 2005
Priority date
Expiry dateMar 17, 2023

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D403/12
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides compounds of formula (I) as well as the use of such compounds in pharmaceutical compositions and methods of treatment.The compounds described herein represent a class of TAFIa inhibitors suitable for use in treating conditions such as thrombosis, atherosclerosis, adhesions, dermal scarring, cancer, fibrotic conditions, inflammatory diseases and those conditions which benefit from maintaining or enhancing bradykinin levels in the body.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.