Patent · US Expired

Pyrrolotriazine inhibitors of kinases

US6982265B1 · kind B1 · utility

64Cited by
6References
9Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 18, 2000
Grant dateJan 3, 2006
Priority date
Expiry dateMay 18, 2020

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides compounds of formula I and pharmaceutically acceptable salts thereof.The formula I compounds inhibit the tyrosine kinase activity of growth factor receptors such as VEGFR-2, FGFR-1, PDGFR, HER-1, HER-2, thereby making them useful as anti-cancer agents. The formula I compounds are also useful for the treatment of other diseases associated with signal transduction pathways operating through growth factor receptors.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.