Patent · US Expired

Substituted diarylamines as MEK inhibitors

US7001905B2 · kind B2 · utility

34Cited by
3References
17Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 12, 2001
Grant dateFeb 21, 2006
Priority date
Expiry dateMar 12, 2021

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C2601/14
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Diarylamines, such as 5-amide substituted diarylamines of formula (I) or formula (II) wherein A is hydroxy, C1-6 alkoxy, or NR6OR7; X is OR12, NR13R12, or NR14; inhibitors of MEK and are useful in the treatment of a variety of proliferative disease states, such as conditions related to the hyperactivity of MEK, as well as diseases modulated by the MEK cascade.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.