Patent · US Expired

Oxazolidinone combinatorial libraries, compositions and methods of preparation

US7002020B1 · kind B1 · utility

1Cited by
1References
7Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 17, 2000
Grant dateFeb 21, 2006
Priority date
Expiry dateJun 25, 2022

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC40B40/00
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Oxazolidinones and methods for their synthesis are provided. Also provided are combinatorial libraries comprising oxazolidinones, and methods to prepare the libraries. Further provided are methods of making biologically active oxazolidinones as well as pharmaceutically acceptable compositions comprising the oxazolidinones. The methods of library preparation include the attachment of oxazolidinones to a solid support. The methods of compound preparation in one embodiment involve the reaction of an iminophosphorane with a carbonyl containing polymeric support.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.