Patent · US Expired

Polymeric drug formulations

US7005454B2 · kind B2 · utility

81Cited by
8References
29Claims
0Family size

Assignee

Inventors

Key dates

Filing dateFeb 24, 1999
Grant dateFeb 28, 2006
Priority date
Expiry dateMay 1, 2021

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K9/7007
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Polymeric drug formulations containing a non-releasing single-phase dispersion of a water-soluble drug in a water-insoluble tissue-compatible polymer matrix. Polymeric drug formulations are also disclosed containing a single-phase dispersion of a water-soluble drug and a water-insoluble tissue-compatible polymer matrix, and a second, phase-disrupting polymer that is non-miscible with the tissue-compatible polymer and is present in an amount sufficient to form phase-separated microdomains of the second polymer in the tissue-compatible polymer matrix, so that the release rate of the water-soluble drug from the tissue-compatible polymer matrix is related to the amount of the second polymer. Methods of preparing the polymeric drug formulations are also described, as well as methods for site-specific drug delivery utilizing the polymeric drug formulations.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.