Patent · US Expired

2-substituted 5-oxazolyl indole compounds useful as IMPDH inhibitors and pharmaceutical compositions comprising same

US7008958B2 · kind B2 · utility

1Cited by

4References

13Claims

0Family size

Assignee

Bristol-Myers Squibb Company · US

Inventors

Scott Hunter Watterson · Pennington, US
T. G. Murali Dhar · Newtown, US
Edwin J. Iwan wicz · Plainsboro, US

Key dates

Filing date	May 20, 2003
Grant date	Mar 7, 2006
Priority date	—
Expiry date	Nov 8, 2023

Classification

Technology area (CPC C)Chemistry; Metallurgy
CPC primaryC07D417/14
WIPO fieldOrganic fine chemistry
WIPO sectorChemistry

Abstract

Compounds having the formula (I), are effective as inhibitors of IMPDH enzyme, wherein R3 is alkyl, substituted alkyl, alkoxy, haloalkoxy, or halogen, preferably methoxy, ethoxy, or trifluoromethoxy; and R1, R2, R4, and R5 are as defined in the specification.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.