Patent · US Expired

Amides that inhibit vanilloid receptor subtype 1 (VR1) receptor

US7037927B2 · kind B2 · utility

1Cited by
1References
7Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 16, 2003
Grant dateMay 2, 2006
Priority date
Expiry dateApr 5, 2024

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D401/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates to compounds of formula (I) that are novel VR1 antagonists useful in treating pain, inflammatory thermal hyperalgesia, urinary incontinence, or bladder overactivity.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.