Patent · US Expired

Butyrylcholinesterase variant polypeptides with increased catalytic efficiency and methods of use

US7049121B2 · kind B2 · utility

15Cited by
13References
10Claims
0Family size

Assignee

Inventors

Key dates

Filing dateDec 20, 2002
Grant dateMay 23, 2006
Priority date
Expiry dateMar 2, 2024

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K38/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention provides twenty-one butyrylcholinesterase variants having increased cocaine hydrolysis activity as well as the corresponding encoding nucleic acids. The invention further provides methods of hydrolyzing a cocaine-based butyrylcholinesterase substrate as well as methods of treating a cocaine-induced condition.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.