Patent · US Expired

CIS-itraconazole crystalline forms and related processes, pharmaceutical compositions and methods

US7078526B2 · kind B2 · utility

14Cited by
22References
16Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 30, 2003
Grant dateJul 18, 2006
Priority date
Expiry dateJan 29, 2024

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D405/14
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The invention provides novel soluble conazole crystalline forms (e.g. itraconazole, posaconazole and saperconazole) that include salts, co-crystals and related solvates useful as pharmaceuticals. The invention also provides pharmaceutical compositions comprising, and processes for making, these conazole crystalline forms. Methods of using such compositions for the treatment or prevention of systemic and local fungal, yeast, and dermatophyte infections are also provided.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.