Patent · US Expired

Naphthalene derivatives, their production and use

US7084149B2 · kind B2 · utility

1Cited by
3References
27Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 22, 2003
Grant dateAug 1, 2006
Priority date
Expiry dateApr 29, 2024

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D401/06
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

A composition containing a compound of the formula:wherein A is a nitrogen-containing heterocyclic group which may be substituted, R1 is a hydrogen atom, hydrocarbon group which may be substituted, or monocyclic aromatic heterocyclic group which may be substituted, R2 is a hydrogen atom or a lower alkyl group which may be substituted, R3, R4, R5, R6, R7, R8 and R9 are independently a hydrogen atom, a hydrocarbon group which may be substituted, a hydroxy group which may be substituted, a thiol group which may be substituted, an amino group which may be substituted, an acyl group or a halogen atom, a salt thereof or a prodrug thereof has steroid C17,20-lyase inhibitory activity, and are useful for preventing and treating a mammal suffering from, for example, primary cancer of malignant tumor, its metastasis and recurrence thereof.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.