Substituted piperidine compounds and methods of their use
US7087749B2 · kind B2 · utility
24Cited by
9References
34Claims
0Family size
Assignee
Inventors
Key dates
| Filing date | Mar 11, 2004 |
| Grant date | Aug 8, 2006 |
| Priority date | — |
| Expiry date | Mar 11, 2024 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D221/06
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
Certain 4-aryl-piperidine compounds, including N-substituted 9β-substituted-5-(3-substituted-phenyl)morphans and N-substituted octahydro-4a-(3-hydroxyphenyl)-10a-methyl-benzo[g]isoquinolines, pharmaceutical compositions, and methods of their use, inter alia, as opioid antagonists are disclosed.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.