Patent · US Expired

Compounds, their use and preparation

US7087750B2 · kind B2 · utility

19Cited by
2References
75Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 22, 2001
Grant dateAug 8, 2006
Priority date
Expiry dateOct 22, 2021

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/08
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The invention provides 2, 3-, 4- or 5-substituted-N1-(arylsulfonyl)indole and (heteroaryl)indole compounds of the general formula (I):in which Ar, R2, R3, R4 and R5 are as defined in the specification. The compounds bind to the 5-HT6 receptor and are useful for the treatment and prophylaxis of disorders mediated by the 5-HT6 receptor, such as obesity and CNS disorders.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.