Patent · US Expired

Bicyclic compounds as inhibitors of chemokine binding to US28

US7101894B2 · kind B2 · utility

0Cited by
9References
4Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 29, 2002
Grant dateSep 5, 2006
Priority date
Expiry dateAug 29, 2022

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D453/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Methods for treating CMV or a CMV-related disease are provided that use compounds having the formula:wherein Ar is a substituted or unsubstituted 5–14 membered heteroaryl group having from 1 to 5 heteroatoms as ring members; R1 is selected from the group consisting of substituted or unsubstituted aryl(C1–C4)alkyl, heteroaryl(C1–C4)alkyl, —C(O)R11, and —C(O)NR11R12, wherein each R11 and R12 independently is substituted or unsubstituted aryl, substituted or unsubstituted aryl(C1–C4)alkyl, substituted or unsubstituted (C4–C8)cycloalkyl(C1–C4)alkyl, substituted or unsubstituted heteroaryl, substituted or unsubstituted heteroaryl(C1–C4)alkyl and substituted or unsubstituted hetero(C4–C8)cycloalkyl(C1–C4)alkyl; R2 is H or (C1–C8)alkyl; and ZN is a substituted or unsubstituted hetero(C6–C10)bicycloalkyl group.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.