Patent · US Expired

Isoxazoline derivatives as inhibitors of matrix metalloproteinases and/or TNF-α converting enzyme

US7125870B2 · kind B2 · utility

1Cited by
5References
28Claims
0Family size

Assignee

Inventors

Key dates

Filing dateOct 30, 2003
Grant dateOct 24, 2006
Priority date
Expiry dateSep 24, 2024

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D413/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present application describes novel isoxazoline of formula I or II:or pharmaceutically acceptable salt or prodrug forms thereof, wherein A, R1, R2, R3, R4, Z, U, X, Y, Za, and n are defined in the present specification, which are useful as inhibitors of matrix metalloproteinases (MMP), TNF-α converting enzyme (TACE), or a combination thereof.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.