Patent · US Expired

Avermectin derivatives

US7144866B2 · kind B2 · utility

0Cited by
15References
8Claims
0Family size

Assignee

Inventors

Key dates

Filing dateAug 8, 2001
Grant dateDec 5, 2006
Priority date
Expiry dateAug 8, 2021

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07H17/08
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Provided is a compound represented by the general formula (I) or a salt thereof:wherein, —XY— represents —CH═CH— and the like, between R2 and the carbon atom at 5-position represents a single bond or a double bond, R1 represents a lower alkyl group, a formyl group, a carboxyl group, a lower alkoxycarbonyl group (wherein a lower alkyl moiety of said lower alkoxycarbonyl group may be substituted with a heterocyclic group) and the like, and R1a represents a hydrogen atom, provided when R1 represents a lower alkoxycarbonyl group and the like, R1a may further represents a lower alkoxycarbonyl group and the like, when between R2 and the carbon atom at 5-position is a single bond, R2 represents a hydroxyl group and the like, and when between R2 and the carbon atom at the 5-position is a double bound, R2 combines with the carbon atom at 5-position to form a hydroxime group (—C(═NOH)) and the like, and R3 represents a hydroxyl group or a tri(lower alkyl)silyloxy group.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.