5-Phenylpyrimidines, methods and intermediate products for the production thereof and use of the same for controlling pathogenic fungi

US7153860B2 · kind B2 · utility

Assignee

• BASF SE

Inventors

• Thomas Grote · Monsheim, DE
• Andreas Gypser · Mannheim, DE
• Joachim Rheinheimer · Ludwigshafen, DE
• Ingo Rose · Mannheim, DE
• Peter Schafer · Ottersheim, DE
• Frank Schieweck · Heßheim, DE
• Hubert Sauter · Mannheim, DE
• Markus Gewehr · Kastellaun, DE
• Bernd Muller · Flintbek, DE
• Jordi Blasco · Hemsbach, DE
• Eberhard Ammermann · Heppenheim, DE
• Siegfried Strathmann · Schifferstadt, DE
• Gisela Lorenz · Neustadt, DE
• Reinhard Stierl · Freinsheim, DE

Key dates

• Filing date: Mar 13, 2002
• Grant date: Dec 26, 2006
• Expiry date: Feb 4, 2023

Classification

• Technology area (CPC C): Chemistry; Metallurgy
• CPC primary: C07D487/04
• WIPO field: Organic fine chemistry
• WIPO sector: Chemistry

Abstract

The invention relates to 5-phenylpyrimidine of formula (I) wherein the substituents have the following designations: R1 represents a five to ten-membered saturated, partially unsaturated or aromatic monocyclic or bicyclic heterocycle which contains between one and four heteroatoms from the group O, N or S, and which can be substituted as defined in the description; R2 represents hydrogen, halogen, cyano, alkyl, halogenalkyl or alkoxy; R3 and R4 represent hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl; together with the nitrogen atom to which they are bonded, R3 and R4 can also form a five or six-membered ring which can be split by a heteroatom and can carry at least one substituent; R5 and R6 represent hydrogen, halogen, alkyl, halogenalkyl or alkoxy; R1 and R8 represent hydrogen, halogen, alkyl or halogenalkyl; and R9 represents hydrogen, halogen, alkyl, alkoxy, cycloalkoxy, halogenalkoxy or alkoxycarbonyl. The invention also relates to methods and intermediate products for producing said compounds and the use of the same for controlling pathogenic fungi