Substituted carboxamides

US7163938B2 · kind B2 · utility

Assignee

• ELI LILLY AND COMPANY · US

Inventors

• David Kent Herron · Indianapolis, US
• Sajan Joseph · Indianapolis, US
• Angela Lynn Marquart · Greenwood, US
• John Joseph Masters · Fishers, US
• David Mendel · Indianapolis, US
• Gerald Floyd Smith · Indianapolis, US
• Philip Waid · Indianapolis, US
• Michael Robert Wiley · Zionsville, US
• Ying Kwong Yee · Kennett Square, US

Key dates

• Filing date: Nov 14, 2001
• Grant date: Jan 16, 2007
• Expiry date: Mar 30, 2022

Classification

• Technology area (CPC C): Chemistry; Metallurgy
• CPC primary: C07D401/14
• WIPO field: Organic fine chemistry
• WIPO sector: Chemistry

Abstract

This application relates to a compound of formula I (or a pharmaceutically acceptable salt thereof) as defined herein, pharmaceutical compositions thereof, and its use as an inhibitor of factor Xa, as well as a process for its preparation and intermediates therefor.