Patent · US Expired

Insulin prodrugs hydrolyzable in vivo to yield peglylated insulin

US7169889B1 · kind B1 · utility

0Cited by
150References
25Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJun 19, 2000
Grant dateJan 30, 2007
Priority date
Expiry dateJun 19, 2020

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61K38/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates generally to hydrolyzable drug-oligomer conjugates, pharmaceutical compositions comprising such conjugates, and to methods for making and using such conjugates and pharmaceutical compositions. For example, a conjugate of insulin, PEG, and oleic acid can be orally administered.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.