Patent · US Expired

Fused heteroaryl derivatives

US7173029B2 · kind B2 · utility

44Cited by
2References
20Claims
0Family size

Assignees

Inventors

Key dates

Filing dateOct 14, 2005
Grant dateFeb 6, 2007
Priority date
Expiry dateOct 14, 2025

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D495/14
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention provides a pharmaceutical composition which is useful as a phosphatidylinositol 3 kinase (PI3K) inhibitor and an antitumor agent, and it provides a novel bicyclic or tricyclic fused heteroaryl derivative or a salt thereof which possesses an excellent PI3K inhibiting activity and cancer cell growth inhibiting activity.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.