Patent · US Expired

Radioactively labelled amino acid analogues, their preparation and use

US7189383B2 · kind B2 · utility

2Cited by
0References
10Claims
0Family size

Assignee

Inventor

Key dates

Filing dateAug 1, 2003
Grant dateMar 13, 2007
Priority date
Expiry dateSep 30, 2023

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P35/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to Halogenated amino acid analogues for use in diagnosis, which compounds have the general formula (I) wherein: R is (C1–C6) alkyl optionally substituted with thioether or ether oxygen atom when n=0, or a substituted aromatic or heteraromatic ring when n=1–6; and m=0 or 1; and X is a halogen atom. The invention further relates to precursor compounds for these analogues, to a method of preparing these analogues, to a pharmaceutical composition comprising these analogues and to the use of these analogues and compositions in the diagnosis of cancer

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.