Substituted arylpyrazines
US7202250B2 · kind B2 · utility
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3References
16Claims
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Inventors
Key dates
| Filing date | Apr 15, 2005 |
| Grant date | Apr 10, 2007 |
| Priority date | — |
| Expiry date | May 20, 2025 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D409/04
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
Arylpyrazine compounds are provided, including arylpyrazines that can bind with high affinity and high selectivity to CRF1 receptors, including human CRF1 receptors. The invention thus includes methods for treatment of disorders and diseases associated with CRF1 receptors, including CNS-related disorders and diseases, particularly affective disorders and diseases, and acute and chronic neurological disorders and diseases.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.