Patent · US Expired

Hydrolytic kinetic resolution of cyclic substrates

US7220870B2 · kind B2 · utility

9Cited by
27References
16Claims
0Family size

Assignee

Inventors

Key dates

Filing dateJan 5, 2005
Grant dateMay 22, 2007
Priority date
Expiry dateJan 5, 2025

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07C2601/16
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The present invention relates to a process for stereoselective or regioselective chemical synthesis which generally comprises reacting a nucleophile and a chiral or prochiral cyclic substrate in the presence of a non-racemic, chiral catalyst to produce a stereoisomerically- and/or regioisomerically-enriched product. The present invention also relates to hydrolytic kinetic resolutions of racemic and diastereomeric mixtures of epoxides.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.