7-amino triazolopyrimidines for controlling harmful fungi

US7307172B2 · kind B2 · utility

Assignee

• BASF SE

Inventors

• Jordi Blasco · Hemsbach, DE
• Hubert Sauter · Mannheim, DE
• Bernd Muller · Flintbek, DE
• Markus Gewehr · Kastellaun, DE
• Wassilios Grammenos · Ludwigshafen, DE
• Thomas Grote · Monsheim, DE
• Andreas Gypser · Mannheim, DE
• Joachim Rheinheimer · Ludwigshafen, DE
• Ingo Rose · Mannheim, DE
• Peter Schafer · Ottersheim, DE
• Frank Schieweck · Heßheim, DE
• Eberhard Ammermann · Heppenheim, DE
• Siegfried Strathmann · Schifferstadt, DE
• Gisela Lorenz · Neustadt, DE
• Reinhard Stierl · Freinsheim, DE
• Günter Krummel · Vendersheim, DE

Key dates

• Filing date: Jul 16, 2002
• Grant date: Dec 11, 2007
• Expiry date: Jul 25, 2023

Classification

• Technology area (CPC A): Human Necessities
• CPC primary: A01N43/90
• WIPO field: Organic fine chemistry
• WIPO sector: Chemistry

Abstract

The invention relates to 7-amino triazolopyrimidines of formula (I), in which the substituents have the following meanings: R1, R2 represent hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, phenyl, naphthyl; or 5-membered or 6-membered heterocyclyl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; or 5-membered or 6-membered heteroaryl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or R1 and R2 can, together with the nitrogen atom, which binds them, form a 5-membered or 6-membered ring containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; R3 represents alkyl, alkenyl, alkynyl, cycloalkyl, phenylalkyl and alkyl halide; whereby R3 and R2 can be unsubstituted or partially or completely substituted according to the description; X represents halogen, cyano, alkoxy, alkyl halide, phenyl or phenyl that is substituted by Ra. The invention also relates to methods and intermediate products for producing said compounds, to agents containing the same, and to their use.