Patent · US Expired

Modulation of KSP kinesin activity with heterocyclic-fused pyrimidinone derivatives

US7332498B2 · kind B2 · utility

19Cited by
90References
10Claims
0Family size

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Key dates

Filing dateNov 23, 2005
Grant dateFeb 19, 2008
Priority date
Expiry dateNov 23, 2025

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D487/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A method of modulating KSP kinesin activity in vitro comprising contacting KSP kinesin with at least one chemical entity chosen from compounds represented by Formula I:and pharmaceutically acceptable salts thereof, where the variables are as defined further herein.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.