Patent · US Expired

Quinolinone derivatives

US7335774B2 · kind B2 · utility

4Cited by
30References
12Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 29, 2005
Grant dateFeb 26, 2008
Priority date
Expiry dateDec 26, 2025

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D471/04
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

A method for synthesizing a 4-amino substituted quinolinone includes reacting a substituted or unsubstituted 2-benzimidazolyl-2-acetate with a substituted or unsubstituted 2-aminobenzonitrile in the presence of a base or an acid. A 4-amino substituted quinolinone compound is formed by the reaction, and the 4-amino substituted quinolinone compound comprises a benzimidazole group.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.