Patent · US Expired

N-(4-(4-methylthiazol-5-yl)pyrimidin-2-yl)-N-phenylamines as antiproliferative compounds

US7388015B2 · kind B2 · utility

6Cited by
1References
25Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 26, 2004
Grant dateJun 17, 2008
Priority date
Expiry dateOct 8, 2024

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P43/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to 2-substituted 4-heteroaryl-pyrimidines, their preparation, pharmaceutical compositions containing them and their use as inhibitors of cyclin-dependent kinases (CDKs) and hence their use in the treatment of proliferative disorders such as cancer, leukaemia, psoriasis and the like.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.