Derivatives of 4-aminopiperidine and their use as a medicament

US7393861B2 · kind B2 · utility

Assignee

• Société de Conseils de Recherches et d'Applications Scientifiques (S.C.R.A.S) SAS · FR

Inventors

• Christophe Thurieau · Paris, FR
• Jerome Gonzalez · Annemasse, FR
• Christophe Moinet · Orvault, FR

Key dates

• Filing date: May 4, 2005
• Grant date: Jul 1, 2008
• Expiry date: Dec 22, 2025

Classification

• Technology area (CPC C): Chemistry; Metallurgy
• CPC primary: C07D417/14
• WIPO field: Pharmaceuticals
• WIPO sector: Chemistry

Abstract

A subject of the present application is new derivatives of 4-aminopiperidines of formulain which R1, R2 and R3 represent various radical, and their preparation processes by synthetic methods in parallel in liquid and solid phase. These products having a good affinity with certain sub-types of somatostatin receptors, they are particularly useful for treating the pathological states or diseases in which one (or more) somatostatin receptors are involved.