Patent · US Expired

Substituted diazabicycloalkane derivatives

US7399765B2 · kind B2 · utility

19Cited by
1References
16Claims
0Family size

Assignee

Inventors

Key dates

Filing dateSep 16, 2004
Grant dateJul 15, 2008
Priority date
Expiry dateNov 2, 2025

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P29/00
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

Compounds of formula (I)Z-Ar1—Ar2  (I)wherein Z is a diazabicyclic amine, Ar1 is a 5- or 6-membered aromatic ring, and Ar2 is selected from the group consisting of an unsubstituted or substituted 5- or 6-membered heteroaryl ring; unsubstituted or substituted bicyclic heteroaryl ring; 3,4-(methylenedioxy)phenyl; carbazolyl; tetrahydrocarbazolyl; naphthyl; and phenyl; wherein the phenyl is substituted with 0, 1, 2, or 3 substituents in the meta- or para-positions. The compounds are useful in treating conditions or disorders prevented by or ameliorated by α7 nAChR ligands. Also disclosed are pharmaceutical compositions comprising compounds of formula (I) and methods for using such compounds and compositions.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.