Antibacterial cyano-(substituted)-methylenepiperidinophenyl oxazolidinones targeting multiple ribonucleoprotein sites

US7405228B2 · kind B2 · utility

Assignee

• Wockhardt Limited · IN

Inventors

• Mahesh Vithalbhai Patel · Aurangabad, IN
• Prasad Keshav Deshpande · Aurangabad, IN
• Milind Dattatraya Sindkhedkar · Aurangabad, IN
• Shrikant Gupte · Aurangabad, IN
• Yati Chugh · Panchkula, IN
• Nitin Shetty · Kalyan-Dombivli, IN
• Milind Shukla · Aurangabad, IN
• Ravindra Dattatraya Yeole · Aurangabad, IN
• Noel De Souza · Mumbai, IN

Key dates

• Filing date: Jul 10, 2003
• Grant date: Jul 29, 2008
• Expiry date: Jul 10, 2023

Classification

• Technology area (CPC C): Chemistry; Metallurgy
• CPC primary: C07D417/14
• WIPO field: Organic fine chemistry
• WIPO sector: Chemistry

Abstract

The present invention provides agents having high antimicrobial activity for preventing and treating infectious diseases. Thus, the present invention provides novel cyano-(substituted)-methylenepiperidinophenyl oxazolidinone derivatives, processes for making the compounds, as well as antimicrobial compositions containing said derivatives as active ingredients and methods of treating bacterial infections with the said derivatives.