N-(heteroaryl)-1H-indole-2-carboxamide derivatives and their use as vanilloid TRPV1 receptor ligands
US7407950B2 · kind B2 · utility
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17Claims
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Key dates
| Filing date | Jun 20, 2007 |
| Grant date | Aug 5, 2008 |
| Priority date | — |
| Expiry date | Jun 20, 2027 |
Classification
- Technology area (CPC C)Chemistry; Metallurgy
- CPC primaryC07D417/12
- WIPO fieldPharmaceuticals
- WIPO sectorChemistry
Abstract
The invention concerns compounds of general formula (I), wherein n, X1, X2, X3, X4, Z1, Z2, Z3, Z4, Z5 and W are as defined herein.Said compounds are ligands of the TRPV1 vanilloid receptor, and are therefore, useful for treating diseases associated with TRPV1 receptors, such as pain and inflammation.
Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.