Patent · US Expired

Cyclosporin analog formulations

US7429562B2 · kind B2 · utility

9Cited by
99References
31Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMar 13, 2006
Grant dateSep 30, 2008
Priority date
Expiry dateMar 13, 2026

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07K7/645
  • WIPO fieldPharmaceuticals
  • WIPO sectorChemistry

Abstract

The present invention relates to formulations containing cyclosporin analogs that are structurally similar to cyclosporin A, in particular isomeric mixtures of cyclosporin analogs that are structurally similar to cyclosporin A. The formulations form stable microemulsion preconcentrates and may provide superior drug bioavailability and/or may reduce one or more adverse effects associated with the administration of cyclosporin. Also disclosed are methods for using and preparing the formulations.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.