Patent · US Expired

Chloromethylation of thiophene

US7462725B2 · kind B2 · utility

1Cited by
2References
8Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 16, 2002
Grant dateDec 9, 2008
Priority date
Expiry dateSep 29, 2024

Classification

  • Technology area (CPC C)Chemistry; Metallurgy
  • CPC primaryC07D333/12
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

The process according to the invention relates to the preparation of 2-chloromethyl-thiophene of the formula (I). During this process thiophene is chloromethylated in the presence of one or more compounds containing keto group and optionally it is transformed into the compound of the formula (II). Compounds of formula (I) and (II) are intermediates of several pharmaceutically active ingredients.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.