Patent · US Active

Conversion process for 2,3-benzodiazepine enantiomers

US7541355B2 · kind B2 · utility

0Cited by
15References
18Claims
0Family size

Assignee

Inventors

Key dates

Filing dateMay 23, 2005
Grant dateJun 2, 2009
Priority date
Expiry dateNov 26, 2026

Classification

  • Technology area (CPC A)Human Necessities
  • CPC primaryA61P25/22
  • WIPO fieldOrganic fine chemistry
  • WIPO sectorChemistry

Abstract

Methods for the racemization of an enantiomer of a 2,3-benzodiazepine molecule into the corresponding racemic mixture under either basic or acidic conditions are described. Furthermore, the invention relates to the conversion of an enantiomer of tofisopam or its metabolites to the corresponding opposite enantiomer.

Source: USPTO / EPO open patent data. Objective bibliographic and citation counts.